Table 3.
PSMA-ligands for PET/CT imaging
Characteristic | [68 Ga]Ga-PSMA-11 | [68 Ga]Ga-PSMA-I&T | [18F]F-DCFPyL | [18F]F-PSMA-1007 | [18F]F-rhPSMA-7.3 |
---|---|---|---|---|---|
Binding motif | Urea-based | Urea-based | Urea-based | Urea-based | Urea-based |
Half-life | 68 min | 68 min | 110 min | 110 min | 110 min |
Dominant excretion route | Kidney | Kidney | Kidney | Liver | Kidney |
Published | 2012 [15] | 2015 [18, 94] | 2011 [14], 2015 [19] | 2016 [20] | 2020 [21] |
Status | Extensive retrospective data; completed phase 2/3; Approved* | Extensive retrospective data | Extensive retrospective data; completed phase 2/3; Approved* | Extensive retrospective data; completed phase 2/3; Approved* | Extensive retrospective data; under phase 3 investigation (NCT04186819 and NCT04186845) |
Characteristics and current status. *Refers to regulatory approval for clinical use and distribution on a national or international level