TABLE 4.
Full library of synthesized [1,2,3]-triazolo [1,5-a] quinoxalin-4(5H)-ones within this work.
| Cmp | [1,2,3]-triazolo [1,5-a] quinoxalin-4(5H)-ones | Yield |
|---|---|---|
| 5a |
|
20% |
| 5b |
|
27% |
| 5c |
|
65% |
| 5d |
|
56% |
| 5e |
|
35% |
| 6 |
|
quantitative |
| 7 |
|
78% |
| 8 |
|
traces |
| 9 |
|
quantitative |
| 10 |
|
86% |
| 11 |
|
quantitative |
| 12 |
|
97% |
| 13 |
|
99% |
| 14 |
|
94% |
| 15 |
|
95% |
| 16 |
|
96% |
| 17 |
|
quantitative |
| 18 |
|
89% |
| 19 |
|
93% |
| 20 |
|
81% |