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. Author manuscript; available in PMC: 2023 Apr 6.
Published in final edited form as: Br J Clin Pharmacol. 2022 Aug 14;88(10):4623–4632. doi: 10.1111/bcp.15477

Table 4.

Simulated steady-state Cabotegravir Trough (Ctrough)1 for extremes of BMI:

CAB Ctrough (ug/mL, Median [90% prediction interval]) for BMI 16.5 kg/m2 (Body weight 43.0kg F; 50.6kg M) CAB Ctrough (ug/mL, Median [90% prediction interval]) for BMI 50 kg/m2 (Body weight 130.6kg F; 153.9kg M)
Male 2.707 [0.931, 5.648] ug/mL 1.102 [0.339, 2.355] ug/mL
Female 3.275 [1.291, 6.676] ug/mL 1.368 [0.527, 2.828] ug/mL
1

For reference: CAB PA-IC90: 0.166 μg/mL; 4*PA-IC90: 0.664 μg/mL; 8*PA-IC90: 1.33 μg/mL