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. 2023 Mar 29;12(7):1038. doi: 10.3390/cells12071038
A ATR inhibitor (ceralasertib)
ABC ATP-binding cassette
ATCC American Type Culture Collection
ATR ataxia telangiectasia and RAD3-related protein
ATRi ATR inhibitor(s)
BRCA1 breast cancer type 1 susceptibility protein
BRCA2 breast cancer type 2 susceptibility protein
BrdU bromodeoxyuridine
C CHK1 inhibitor (MK-8776)
CDI coefficient of drug interaction
CHK1 checkpoint kinase 1
CHK1i CHK1 inhibitor(s)
DDR DNA damage response
DSB double-strand break
ECACC The European Collection of Authenticated Cell Cultures
HGSOC high-grade serous ovarian cancer
HI-FBS heat-inactivated fetal bovine serum
IC50 concentration of drug required to reduce cell viability to 50%
MDR multidrug resistance
MDR1 multidrug resistance protein 1
MDRi multidrug resistance inhibitor(s)
MFI geometric mean fluorescence intensity
NGS next-generation sequencing
NHEJ non-homologous end joining
O olaparib
OC ovarian cancer
ORF open reading frame
PARG poly(ADP-ribose) glycohydrolase
PARP1 poly(ADP-ribose) polymerase 1
PARPi PARP inhibitor(s)
PDT population doubling time
PEO1-OR PEO1 olaparib-resistant cell line
QCI-IT Qiagen Clinical Insight Interpret Translational
SF surviving fraction
Tar tariquidar
WES whole-exome sequencing