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. 2023 Apr 20;13(4):698. doi: 10.3390/biom13040698
3α5βP 5β-pregnan-3α-ol-20-one
c ratio of the equilibrium dissociation constant in the active state to that in the resting state (a measure of efficacy)
ΔG free energy change
GABA γ-aminobutyric acid
GABAA γ-aminobutyric acid type A
KR equilibrium dissociation constant of a compound in the resting receptor
NS-1738 N-(5-Cl-2-hydroxyphenyl)-N′-[2-Cl-5-(trifluoromethyl)phenyl]-urea
PA probability of being in the active state;
PAM positive allosteric modulator
PAM-2 (E)-3-(furan-2-yl)-N-(p-tolyl)-acrylamide.