| 3α5βP | 5β-pregnan-3α-ol-20-one |
| c | ratio of the equilibrium dissociation constant in the active state to that in the resting state (a measure of efficacy) |
| ΔG | free energy change |
| GABA | γ-aminobutyric acid |
| GABAA | γ-aminobutyric acid type A |
| KR | equilibrium dissociation constant of a compound in the resting receptor |
| NS-1738 | N-(5-Cl-2-hydroxyphenyl)-N′-[2-Cl-5-(trifluoromethyl)phenyl]-urea |
| PA | probability of being in the active state; |
| PAM | positive allosteric modulator |
| PAM-2 | (E)-3-(furan-2-yl)-N-(p-tolyl)-acrylamide. |