Table 2.
Results of direct fluorescence anisotropy titrations with ExoI and RecO. IC50 values are shown for comparison.
mSSB | IC50 on ExoI (µM) | EC50 on ExoI (µM) | IC50 on RecO (µM) | EC50 on RecO (µM) |
---|---|---|---|---|
F-wtSSB | 4.54 ± 0.34 | 0.35 ± 0.04 | 4.66± 0.24 | 0.37 ± 0.03 |
F-4Cl-Phe2 | 0.56 ± 0.03 | 0.15 ± 0.02 | 0.41 ± 0.27 | 0.26 ± 0.01 |
F-4F-Phe2 | 1.93 ± 0.81 | 0.36 ± 0.03 | 0.52 ± 0.28 | 0.23 ± 0.02 |
F-4CF3-Phe2 | 0.33 ± 0.02 | 0.04 ± 0.002 | 0.56 ± 0.42 | 0.18 ± 0.03 |
F-NM-Asp3 | 3.88 ± 0.13 | 0.86 ± 0.11 | 1.88 ± 0.09 | 0.27 ± 0.04 |
F-Glu5 | 1.49 ± 0.10 | 0.11 ± 0.01 | 1.41 ± 0.55 | 0.20 ± 0.02 |
F-Leu6 | 0.92 ± 0.06 | 0.20 ± 0.03 | 3.23 ± 0.16 | 0.31 ± 0.03 |
F-nLe6 | 2.68 ± 0.54 | 0.20 ± 0.01 | 9.36 ± 0.08 | 0.20 ± 0.01 |
F-Pip7 | 0.89 ± 0.14 | 0.09 ± 0.01 | 3.31 ± 0.44 | 0.25 ± 0.03 |
F-3Cl-Phe8 | 3.40 ± 2.41 | 0.25 ± 0.02 | 0.36 ± 0.04 | 0.22 ± 0.03 |
F-4CF3-Phe8 | 0.39 ± 0.07 | 0.09 ± 0.01 | 5.97 ± 2.43 | 0.26 ± 0.02 |