Table 1.

3-Amino-1,2,4-triazine derivatives 4a–j, 5a–j and their relative yields.

Cpd	R	R1	Overall Yield%	4 (%) 5 (%)	Cpd	R	R1	Overall Yield%	4 (%) 5 (%)
4a	H	H	80	42	4f	Br	Cl	79	40
5a				38	5f				39
4b	Br	H	86	44	4g	H	F	81	41
5b				42	5g				40
4c	H	Br	94	49	4h	Br	F	85	43
5c				45	5h				42
4d	Br	Br	92	48	4i	H	OCH3	84	47
5d				44	5i				37
4e	H	Cl	87	46	4j	Br	OCH3	96	48
5e				41	5j				48