Table 2. In Vitro TS Activitya.
| compounds | IC50 (μM) |
|---|---|
| 8 | 3.67 ± 0.58 |
| 9 | 1.01±0.41 |
| 10 | 1.25 ± 0.35 |
| 12 | 2.93 ± 0.71 |
| 15 | 2.57 ± 0.31 |
| 17 | 0.81±0.21 |
| pemetrexed | 2.81 ± 0.31 |
IC50 values are the mean ± S.D. of three separate experiments.
| compounds | IC50 (μM) |
|---|---|
| 8 | 3.67 ± 0.58 |
| 9 | 1.01±0.41 |
| 10 | 1.25 ± 0.35 |
| 12 | 2.93 ± 0.71 |
| 15 | 2.57 ± 0.31 |
| 17 | 0.81±0.21 |
| pemetrexed | 2.81 ± 0.31 |
IC50 values are the mean ± S.D. of three separate experiments.