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. 2023 Jun 3:1–7. Online ahead of print. doi: 10.1007/s00044-023-03079-x

Table 2.

SAR studies: effect of varying the amino side chain

graphic file with name 44_2023_3079_Tabn_HTML.gif
Compound R IC50a nM (±SD)
18 graphic file with name 44_2023_3079_Tabo_HTML.gif 21 (±3.1)
20 graphic file with name 44_2023_3079_Tabp_HTML.gif 4200 (±280)
21 graphic file with name 44_2023_3079_Tabq_HTML.gif 12 (±9.8)
22 graphic file with name 44_2023_3079_Tabr_HTML.gif 90 (±49)
23 graphic file with name 44_2023_3079_Tabs_HTML.gif 99 (±31)
24 graphic file with name 44_2023_3079_Tabt_HTML.gif 220 (±93)
25 graphic file with name 44_2023_3079_Tabu_HTML.gif 23 (±1.4)
26 graphic file with name 44_2023_3079_Tabv_HTML.gif 220 (±110)

aAAK1 IC50 values are means of two or more experiments, standard deviation is given in parentheses