Table 2.
The biodistribution of [18F]AlF-NOTA-ADH-1 in PDX xenograft model( ± SD, %ID/g.).
| Organs | Non-blocking group | Blocking group | |||
|---|---|---|---|---|---|
| 30min | 60min | 90min | 120min | 60min | |
| Blood | 0.69±0.22 | 0.40±0.18 | 0.39±0.11 | 0.41±0.07 | 0.35±0.14 |
| Brain | 0.62±0.14 | 0.99±0.47 | 0.63±0.18 | 0.51±0.27 | 0.86±0.21 |
| Heart | 2.54±0.97 | 0.96±0.17 | 0.95±0.25 | 0.81±0.28 | 0.82±0.02 |
| Lung | 4.38±1.33 | 3.41±0.44 | 3.52±1.76 | 2.07±0.94 | 2.37±0.14 |
| Liver | 12.28±1.23 | 11.31±2.30 | 10.43±1.97 | 9.20±1.66 | 10.35±1.15 |
| Spleen | 1.81±0.48 | 1.41±0.24 | 1.13±0.03 | 0.86±0.25 | 1.25±0.20 |
| Kidney | 17.75±5.89 | 15.82±1.17 | 12.50±0.89 | 8.52±2.09 | 11.62±2.40 |
| Stomach | 3.23±1.69 | 3.40±0.12 | 6.16±1.58 | 1.60±1.04 | 2.24±0.16 |
| Intestines | 3.82±0.12 | 2.14±0.04 | 3.93±2.67 | 2.53±2.00 | 2.49±0.33 |
| Muscle | 1.41±0.20 | 1.56±0.07 | 2.03±0.05 | 1.18±0.60 | 1.68±0.06 |
| Bone | 1.74±0.81 | 2.29±0.96 | 1.65±1.30 | 0.74±0.35 | 2.16±0.09 |
| Skin | 0.11±0.04 | 0.95±0.46 | 1.51±0.02 | 1.56±0.66 | 0.54±0.14 |
| Tumor | 8.04±1.82 | 10.76±2.16 | 7.18±0.53 | 4.93±1.65 | 3.75±0.07 |
| T/Blood | 10.72± 1.02 | 19.21± 2.20 | 13.54± 0.35 | 10.27±1.36 | 9.39± 0.10 |
| T/Muscle | 5.69±0.72 | 8.70±2.68 | 4.15±1.86 | 3.97±1.56 | 2.12±0.06 |