Table 4.
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Conditions: 1 (0.1 mmol, 1.0 equiv), methyl 4-iodobenzoate (2.0 equiv), Pd(OAc)2 (10 mol%), TDG (30 mol%), L12 (60 mol%), AgTFA (3.0 equiv) and ClCH2COOH (1.0 equiv) in HFIP (0. 5 mL), 120°C, under air, 12 h.
Yield and ratio determined by 1H NMR of the crude mixture.
Reaction time: 48h.