Table 1.
Evaluation of effect of different zinc-binding groups on HDAC inhibitory activity by growth inhibition assay using HCT116 cells at a maximum concentration of 100 μM.
Compound | HCT116 IC50 | Compound | HCT116 IC50 |
---|---|---|---|
| |||
![]() |
>100 |
![]() |
>100 |
![]() |
>100 |
![]() |
>100 |
![]() |
>100 |
![]() |
>100 |
![]() |
>100 |
![]() |
>100 |
![]() |
>100 |
![]() |
>100 |
![]() |
>100 |
![]() |
>100 |
![]() |
>100 |
![]() |
>100 |
![]() |
>100 |
![]() |
54.39 ± 6.02 |
![]() |
>100 |