Table 2. Pyrrolocarbazole Analogues (XVII)a.
comp | R | R1 | R2 | IC50 (nM) |
---|---|---|---|---|
44 | H | Ph | H | 130 |
45 | H | 2-Cl Bn | H | 11 |
46 | H | 2,6-diCl Bn | H | 28 |
47 | H | 2-Cl Bn | (CH2)3OH | 9 |
48 | H | 2-Cl Bn | (CH2)2CONH2 | 6 |
49 | (CH2)4NMe2 | 2-Cl Bn | H | 49 |
50 | O(CH2)3Nmorph | 2-Cl Bn | (CH2)2OH | 15 |
Bn stands for benzene, Ph for phenyl, and morph for morpholine.