Table 1. TC50 of Tested Compounds on A549, H1299, H1975, and MRC-5 Cellsa.
| TC50 (μM) |
||||
|---|---|---|---|---|
| compound | A549 | H1299 | H1975 | MRC-5 |
| 3 | 22 ± 1.0 | 27 ± 0.8 | 28 ± 2.0 | 45 ± 8.0 |
| 4a | 13 ± 0.3 | 13 ± 0.1 | 23 ± 2.0 | 17 ± 3.0 |
| 4b | 17 ± 0.5 | 17 ± 0.3 | 35 ± 4.0 | |
| 5a | 32 ± 0.9 | 33 ± 0.7 | 33 ± 2.0 | |
| 5b | 19 ± 0.4 | 16 ± 0.6 | 25 ± 5.0 | |
| 5c | 11 ± 0.5 | 11 ± 0.3 | 15 ± 1.0 | 17 ± 0.3 |
| 5d | 16 ± 0.4 | 18 ± 0.5 | 29 ± 4.0 | |
| regorafenib | 13 ± 0.8 | 10 ± 0.4 | 16 ± 0.5 | 18 ± 2.0 |
| Leflunomide | 100 < TC50 <300 | 300 < | 100 < | 300 < |
All values are expressed as mean ± standard error (n = 6).