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. 2023 Jun 8;8(24):21769–21780. doi: 10.1021/acsomega.3c01323

Table 1. TC50 of Tested Compounds on A549, H1299, H1975, and MRC-5 Cellsa.

  TC50 (μM)
 
compound A549 H1299 H1975 MRC-5
3 22 ± 1.0 27 ± 0.8 28 ± 2.0 45 ± 8.0
4a 13 ± 0.3 13 ± 0.1 23 ± 2.0 17 ± 3.0
4b 17 ± 0.5 17 ± 0.3 35 ± 4.0  
5a 32 ± 0.9 33 ± 0.7 33 ± 2.0  
5b 19 ± 0.4 16 ± 0.6 25 ± 5.0  
5c 11 ± 0.5 11 ± 0.3 15 ± 1.0 17 ± 0.3
5d 16 ± 0.4 18 ± 0.5 29 ± 4.0  
regorafenib 13 ± 0.8 10 ± 0.4 16 ± 0.5 18 ± 2.0
Leflunomide 100 < TC50 <300 300 < 100 < 300 <
a

All values are expressed as mean ± standard error (n = 6).