Table 4. Phase II Stability in Liver Microsomes of Dim22 and Standards.
human |
mouse |
|||||||
---|---|---|---|---|---|---|---|---|
compound | Cli | SD | ![]() |
SD | Cli | SD | ![]() |
SD |
μL/min/mg protein | min | μL/min/mg protein | min | |||||
Dim22 | 51.5 | 0.7 | 26.9 | 0.4 | 57.0 | 2.7 | 24.3 | 1.1 |
7-EC | 46.1 | 0.4 | 30.0 | 0.2 | 290.9 | 105.4 | 5.1 | 1.8 |
7-OHC | 390.0 | 53.1 | 3.6 | 0.5 | 533.3 | 105.0 | 2.7 | 0.5 |