Official websites use .gov
A
.gov website belongs to an official
government organization in the United States.
Secure .gov websites use HTTPS
A lock (
) or https:// means you've safely
connected to the .gov website. Share sensitive
information only on official, secure websites.
Cytostatic activity of peptide/drug conjugates on EBC-1.
| Conjugate | IC50 ± SD (µM) * |
|---|---|
| EBC-1 | |
| Dabcyl-Cys-(Arg)6-Cys-(Gly)4-Lys(DauSuc) orto BBMB | 17.8 ± 2.2 |
| Dabcyl-Cys-(Arg)6-Cys-(Gly)4-Lys(DauSuc) para BBMB | 19.8 ± 0.1 |
* The cells were incubated with the compound for 3 h, and subsequently cultured in a serum-containing medium for three days. The IC50 values were determined by Alamar-blue assay as described in the text. Standard deviation values (SD) are also presented.
