Table 5.
Metabolism and excretion parameters of compounds 3c, 3e, 3g, 3h, 3l, and mxm (meloxicam).
| Parameter | Compound | |||||
|---|---|---|---|---|---|---|
| 3c | 3e | 3g | 3h | 3l | mxm | |
| CYP1A2 inhibitor | No | No | No | No | No | No | 
| CYP2C19 inhibitor | Yes | Yes | Yes | Yes | No | No | 
| CYP2C9 inhibitor | Yes | Yes | Yes | Yes | No | Yes | 
| CYP2D6 inhibitor | No | Yes | Yes | No | Yes | No | 
| CYP3A4 inhibitor | Yes | Yes | Yes | Yes | No | No |