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. 2023 Apr 20;114(7):2699–2708. doi: 10.1111/cas.15803

TABLE 2.

Inhibitors targeting autophagy‐related factors.

Targeted ATG Compound IC50 Reference
ULK1/ULK2 SBI‐0206965 108 nM/711 nM 69
MRT67307 45 nM/38 nM 70
MRT68921 2.9 nM/1.1 nM
Compound 6 8 nM/− 71
ULK‐100 1.6 nM/2.6 nM 72
ULK‐101 8.3 nM/30 nM
VPS34 SAR405 1.2 nM 73
VPS34‐IN1 25 nM 74
PIK‐III 18 nM 75
Compound 31 2 nM 76
SB02024 14 nM 77
ATG7 Compound 18 48 nM 78
Compound 19 52 nM
Compound 37 62 nM
Atg4A/Atg4B NSC185058 −/50 μM 79
Tioconazol 1.3 μM/1.8 μM 80
LV320 35.5 μM/24.5 μM 81
S130 7.11 μM/3.24 μM 82
FMK‐9a −/80 nM 83
UAMC‐2526 −/− 84
ATG4B‐LC3 PPI SUPR4B1W 120 nM (KD) 85
ATG5‐ATG16L1 PPI Peptide 10 12 nM (KD) 86
Beclin1‐ATG14L PPI Cmpound 19 33.9 uM 87

Note: (−): not applicable, not available.