Table 4.
RT inhibitory activity of some selected compounds.
| Compd. | R10L2 | R10L4 | R13L2 | IAS-0 | EFVb |
|---|---|---|---|---|---|
| IC50 (μmol/L)a | 0.060 ± 0.009 | 0.070 ± 0.009 | 0.057 ± 0.012 | 0.018 ± 0.002 | 0.030 ± 0.000 |
IC50: Compound concentration required to inhibit 50% incorporation of biotin-labeled UTP by HIV-1 (WT) RT.
All data were obtained from one batch with the same method.