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. 2023 Jun 24;64:102793. doi: 10.1016/j.redox.2023.102793

Table 1.

The Keap1-Nrf2 binding affinity of the unsymmetric bisulfonamides determined by the fluorescence anisotropy assay.Image 1.

Entry R KD (nM)a Entry R KD (nM)
A1 Image 2 >10000 A7 Image 3 1433
A2 Image 4 1304 A8 Image 5 1153
A3 Image 6 >10000 A9 Image 7 1143
A4 Image 8 1109 A10 Image 9 3270
A5 Image 10 >10000 A11 Image 11 1275
A6 Image 12 2066 A12 Image 13 >10000
POZL Image 14 940 A13 Image 15 >10000
NXPZ-2 Image 16 230
a

Duplicated experiment and the average data.