Table 2. . TAS-117 dose-escalation levels.
| Dose levels | TAS-117 dose | |
|---|---|---|
| QD regimen, mg/day | Intermittent dosing (4 days on/3 days off per week), mg/day | |
| -1 | 12 | 20 |
| 1 | 16 | 24 |
| 2 | 20 | 28 |
| 3 | 24 | 32 |
QD: Once daily.
| Dose levels | TAS-117 dose | |
|---|---|---|
| QD regimen, mg/day | Intermittent dosing (4 days on/3 days off per week), mg/day | |
| -1 | 12 | 20 |
| 1 | 16 | 24 |
| 2 | 20 | 28 |
| 3 | 24 | 32 |
QD: Once daily.