Skip to main content
[Preprint]. 2023 Jul 4:2023.07.04.547721. [Version 1] doi: 10.1101/2023.07.04.547721

Table 1.

C10-S66K Binding Affinities

Synthetic Opioid KD (M)
Carfentanil 6.899E-11
Fentanyl 2.277E-10
Acetylfentanyl 1.903E-10
Butyrylfentanyl 1.323E-10
p-Tolylfentanyl 1.781E-10
3-Methylfentanyl 8.809E-09
α-Methylfentanyl 7.102E-10
Sufentanil 1.909E-08
Alfentanil >10 μM
Remifentanil >1 μM
Naloxone No binding