Table 5. Effective Concentrations of MARK4 Inhibitors Causing 50% Loss of Cell Viability (EC50 Values) in HeLa and U87MG Cancer Cell Linesa.
EC50 (μM) |
|||||
---|---|---|---|---|---|
compound | HeLa | U87MG | MDA-MB-435 | U251 | HGFs |
23a | 2.13 ± 0.08 | 4.13 ± 0.06 | 1.76 ± 0.06 | 7.98 ± 0.21 | 3.55 ± 0.08 |
23b | 2.52 ± 0.07 | 4.22 ± 0.12 | ND | ND | ND |
23c | 2.16 ± 0.03 | 3.51 ± 0.09 | ND | ND | ND |
16a | >50 | >50 | >50 | >50 | >50 |
16b | >50 | >50 | ND | ND | ND |
16c | >50 | >50 | ND | ND | ND |
Results are presented as mean ± SE of three independent experiments. ND = Not determined.