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. 2018 Dec 18;10(1):24–35. doi: 10.1007/s12672-018-0353-6

Table 3.

Cell-based binding assay

Compound % competition of [3H] MB binding1
[3H] MB 82
SPEP-5 57
SPEP-10 67
SPEP-19 82
SPEP-22 85
SPEP-24 90
SPEP-26 73
SPEP-27 71
SPEP-36 91
SPEP-41 50
SPEP-42 31
SPEP-43 73
HGSF-1 10
HGSF-2 40

1Percent inhibition of MB binding in cultured cell (2080 genital skin fibroblast, GSF) assay; conjugate concentration 500 nM, except for SPEP-24, which was at 50 nM