Table 2. Whole-Cell Target-Based Screena.
MIC (μg/mL) |
||||
---|---|---|---|---|
Mtb strains | 22 | 23 | 11 | streptomycin |
H37Rv | 1 | 0.3 | 0.25 | 0.25 |
TB71 | 0.25 | 0.03–0.06 | 0.125 | 0.25 |
TB173 Pi [25 ng/mL] | 0.125 | 0.06 | 0.125 | 0.25 |
TB173 Pi [15 ng/mL] | 0.125 | 0.01 | 0.125 | 0.25 |
Activity of 22 and its derivatives against Mtb H37Rv, parental TB71, and conditional mutant TB173 strains (determined by REMA).