Table 2.
Commonly used drugs and targets for endocrine therapy of breast cancer.
Type | Drugs | Target |
---|---|---|
Anti-estrogens | Tamoxifen, toremifene, raloxifene, fulvestrant | ER |
Aromatase inhibitor | Anastrozole, letrozole, exemestane | Aromatase enzymes |
LHRH analogues | Goserelin, leuprorelin, triptorelin | LHRH receptor |
Progestogens | Megestrol | PR |
CDK4/6 inhibitor | Palbociclib, ribociclib, abemaciclib, trilaciclib | CDK4、CDK6 |