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. 2023 Jul 7;13:1218206. doi: 10.3389/fonc.2023.1218206

Table 2.

Commonly used drugs and targets for endocrine therapy of breast cancer.

Type Drugs Target
Anti-estrogens Tamoxifen, toremifene, raloxifene, fulvestrant ER
Aromatase inhibitor Anastrozole, letrozole, exemestane Aromatase enzymes
LHRH analogues Goserelin, leuprorelin, triptorelin LHRH receptor
Progestogens Megestrol PR
CDK4/6 inhibitor Palbociclib, ribociclib, abemaciclib, trilaciclib CDK4、CDK6