Table 2.
Mean Pharmacokinetic Parameters of Tirzepatide in Female Sprague Dawley Rats Following a Single Subcutaneous Administration.
Dose | Tmax | Cmax | AUC0–96 | T1/2 | CL/F |
---|---|---|---|---|---|
nmol/kg | (hr) | (nmol/L) | (hr*nmol/L) | (hr) | (mL/hr/kg) |
31 | 12 | 127 | 3742 | 9.3 | 8.31 |
104 | 12 | 310 | 10040 | 10.3 | 10.3 |
Abbreviations: AUC0–96hr = area under the plasma concentration versus time curve from 0 to 96 hours, Cmax = maximum plasma concentration, Tmax = time of Cmax, T1/2 = half-life, CL/F = clearance.