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. 2023 Jul 11;8(29):25903–25923. doi: 10.1021/acsomega.3c01682

Table 5. AlkP Activity after an Incubation of 72 h in Ishikawa Cells.

  1 nM 10 nM 100 nM 1 μM 10 μM
E2 n.d.b 6.86 ± 0.69a n.d. n.d. n.d.
Tam n.d. n.d. n.d. 1.60 ± 0.55 1.02 ± 0.37
OH-Tam n.d. n.d. n.d. 1.73 ± 0.46 0.60 ± 0.20
2B 1.36 ± 0.97 1.47 ± 0.45 1.86 ± 0.73 2.01 ± 0.55a 0.04 ± 0.07
2C 1.18 ± 0.67 1.32 ± 0.25 1.73 ± 0.71 1.89 ± 0.45a 0.00 ± 0.00
4 n.d. n.d. 3.91 ± 1.40 3.76 ± 1.41 n.d.
a

Solvent control (DMSO) was set to 1; p < 0.05 (Tukey’s test).

b

n.d. = not determined.