Table 1.
IC50 and EC50 values for UNbC5-1, UNbC5-2, Ecu-mab, and RaCI3 for inhibiting complement activity and binding complement C5
Inhibitor | IC50 (nM) CP | EC50 (nM) C5 WT | EC50 (nM) C5 R885H |
---|---|---|---|
UNbC5-1 | 137 ± 83 | 0.38 ± 0.20 | 1.5 ± 0.4 |
UNbC5-2 | 24 ± 15 | 0.12 ± 0.01 | 22.4 ± 17.0 |
Ecu-mab | 9 ± 4 | 0.05 ± 0.01 | ND |
RaCI3 | 42 ± 8 | - | - |
Binding and inhibition curves were fitted using the GraphPad Prism 9.3.0 function “[inhibitor] versus normalized response–variable slope” & “Asymmetrical Sigmoidal, 5PL, X is concentration”. IC50 and EC50 values were calculated for three individual experiments using the fitted curves, and SD were determined.