Stuctures and Reported Potencya
of Representative P2Y14R Antagonists, Derived from Lead Piperidine 1 (Including C-Bridged 2 and Uncharged 3 Bioisosteres) and Recently Reported 2-Phenyl-benzoxazole Acetamide 4a and 5-Amido-1H-pyrazole-3-carboxylic Acid 4b Derivatives 20,21
bInhibitory activity in a cAMP assay.16,20aIC50 in a fluorescent binding assay, unless noted.