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. 2022 May 20;53(3):457–465. [Article in Chinese] doi: 10.12182/20220560208

表 3. The screening of WRAP53β co-inhibitory drugs.

WRAP53β共抑制药物筛选

Database Drug Targeted gene t P
 CGP: Cancer genome project; CTRP: The cancer therapeutics response portal; ATM: Ataxia telangiectasia-mutated gene; CDK1: Cyclin-dependent kinase 1; MDM4: Murine double minute 4; TERT: Telomerase reverse transcriptase.
CGP CP-466722 ATM 5.20 0.00
AT7519 CDK1 4.02 0.00
PHA-793887 CDK1 5.40 0.00
58131-57-0 MDM4 4.19 0.00
CTRP KU-55933 ATM 2.58 0.01
KU-60019 ATM 2.61 0.01
Telomerase inhibitor Ⅸ TERT 3.06 0.00