Recommended dosage for older adults | 0.125–0.25 mg [25] |
Indications | Sleep onset insomnia, short-term use [25, 26•• |
Contraindications | Hypersensitivity to triazolam or other benzodiazepines; contraindicated in women who are pregnant or may become pregnant; medications that impair the oxidative metabolism mediated by P4503A (CYP3A) [28, 29] |
Main drug interactions | Opioids; drugs that inhibit triazolam metabolism via cytochrome P4503A; drugs and other substances demonstrated to be CYP3A inhibitors; drugs that affect triazolam pharmacokinetics by other mechanisms including ranitidine [29] |
Main side effects | Drowsiness; headache; dizziness; light headedness; “pins and needles” sensations on skin; coordination difficulties [29] |