TABLE 12.

Additional and less potent inhibitors of AEA cellular uptake relative to inhibition of AEA degradation (by FAAH) or intracellular transport (by FABP5)

Compound	AEA Cellular Uptake Inhibition
	IC50 (µM)	Cell Type	FAAH IC50 Value (µM)	FABP5 Ki Value (µM)
BMS309403 Sulsky et al., 2007; Kaczocha et al., 2009; Berger et al., 2012; Kaczocha et al., 2012; Nicolussi et al., 2014a	∼100 [57% inh.] >100 [48% inh.] 24.7 >100 [30% inh.]	N18TG2 COS7-FAAH-eGFP U937 HMC-1*	>100 >100	0.35 0.75 0.89
SBFI-26 (RT26) Berger et al., 2012: Zhou et al., 2019a	∼20 [40% inh.]	HeLaa	>50	0.9

^aCells lacking FAAH-activity.