Table 2.
The inhibition at 50 μM ligand concentration afforded by compounds 1 and 12–14.
| Compound | Structure | Inhibition (%) at 50 μM |
|---|---|---|
| 1 |
|
> 90 |
| 12 |
|
16 ± 1 |
| 13 |
|
< 10 |
| 14 |
|
14 ± 1 |
The inhibition at 50 μM ligand concentration afforded by compounds 1 and 12–14.
| Compound | Structure | Inhibition (%) at 50 μM |
|---|---|---|
| 1 |
|
> 90 |
| 12 |
|
16 ± 1 |
| 13 |
|
< 10 |
| 14 |
|
14 ± 1 |