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. 2023 Aug 22;16(9):1191. doi: 10.3390/ph16091191

Table 1.

Summary of proposed targets of BIM compounds used as standards [41,59,65,68,69,70,71,72,73,74,75].

BIM Proposed Targets
BIM-I PKC, GSK-3β, 5-HT3, ABCG2, OCT-1, PDK1, MSK1, MAPKAP-K1, S6K1, Chk1, PKA, DYRK1
BIM-II PKC, ABCG2, OCT-1, PDK1, MSK1, MAPKAP-K1, PKA, DYRK1
BIM-III PKC, ABCG2, OCT-1, S6K1, MAPKAPK1, RSK2, MSK1, PDK1
BIM-IV PKC, PKA, MAPKAPK1, MSK1, ABCG2
BIM-V ABCG2, SK6
BIM-VI OCT-1
BIM-VII OCT-1
BIM-VIII PKC, GSK-3β, carbachol-evoked noradrenaline release, OCT-1, PDK1, MSK1, S6K1, PKA, DYRK1, MAPKAPK1
BIM-IX PKC, GSK-3β, MAPKAPK1, MSK1, OCT-1, S6K1
BIM-X Multiple Protein Kinases
BIM-XI PKC, T-cell activation