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. 2023 Sep 26;10(3):37–60. doi: 10.15586/jkcvhl.v10i3.295

Table 1:

Grouped histology.

Agent (trial, year) Phase N per group Histology (%) Primary endpoint ORR, % (95% CI) mPFS, months
(95% CI)
OS, months
(95% CI)
Sunitinib (2012)(17) II 31 22 (71) papillary
3 (10) chromophobe
5 (16) unclassified
1 (3) Xp11.2 translocation
ORR 35 (19–52) 6.4 (4.2–8.6) NR, estimated at 25.6 (8.4–42.9)
1-year OS: 65%
Sunitinib vs. everolimus
(ESPEN, 2016)(18)
II 33 Sunitinib
35 Everolimus
14 (43) papillary
6 (18) chromophobe
4 (12) unclassified
3 (9) translocation unspecified
6 (18) clear cell with sarcomatoid features
13 (38) papillary
6 (17) chromophobe
6 (17) unclassified
4 (11) translocation unspecified
6 (17) clear cell with sarcomatoid features
PFS 9
2.8
6.1
4.1 (P = 0.6)
16.2
14.9 (P = 0.18)
Sunitinib vs. everolimus
(ASPEN, 2016)(19)
II 51 Sunitinib
57 Everolimus
33 (65) papillary
10 (20) chromophobe
8 (16) unclassified
37 (65) papillary
6 (10) chromophobe
14 (25) unclassified
PFS 18
9
8.3 (8.0–11.4)
5.6 (5.0–5.6)
HR: 1.41 (0.03–1.92)
31.5 (14.8–NA)
13.2 (9.7–37.9)
HR: 1.12 (0.7–2.1)
Temsirolimus vs. sunitinib (CESAR, 2020)(20) II 12 Temsirolimus
10 Sunitinib
8 (67) papillary
2 (17) chromophobe
1 (8) medullary
1 (8) unclassified
8 (80) papillary
2 (20) unclassified
PFS NA
NA
9.3
13.2
HR: 1.64 (0.65–4.18)
19.4
19.8
Pazopanib
(2018)(22)
II 29 19 (66) papillary
3 (10) chromophobe
7 (24) unclassified
ORR 28 16.5 (10.9–22.1) NR
Axitinib (2018)(23) II 40 26 (60) papillary
4 (10) chromophobe
7 (18) MiT translocation
3 (7) others
PFS 37.5 7.4 (5.2–9.5) 12.1 (6.4–17.7)
Everolimus + bevacizumab (2016)(24) II 34 5 (14) papillary
5 (14) chromophobe
2 (6) medullary
23 (66) unclassified
PFS 29 11 (3.8–19.3) 18.5
Everolimus + bevacizumab (2020)(25) II 37 13 (35) papillary
1 (3) translocation unspecified
23 (62) unclassified
PFS 35 13.7 (10.8–16.4) 33.9 (23.3–71.9)
Nivolumab
(Checkmate 374, 2020)(26)
IIIb/IV 44 24 (55) papillary
7 (16) chromophobe
1 (2) medullary
1 (2) collecting duct
2 (5) translocation unspecified
8 (18) unclassified
1 (2) unreported
High-grade immune-mediated adverse events 13.6 (5.3–27.4) 2.2 (1.8–5.4) 16.3 (9.2–NE)
Atezolizumab + bevacizumab (2020)(27) II 42 12 (35) papillary
10 (29) chromophobe
1 (3) medullary
5 (15) collecting duct
5 (15) TFE3translocation
9 (26) unclassified
ORR 26 8.3 months (5.7–10.9) NR
Cabozantinib + atezolizumab
(COSMIC,
2021)(29)
Ib 32 15 (47) papillary
9 (28) chromophobe
1 (3) collecting duct
1 (3) fumarate-hydrase deficient
1 (3) MiT-family translocation
1 (3) translocation unspecified
1 (3) poorly differentiated
1 (3) spindle-cell
1 (3) clear cell
ORR 31 (20–44) 9.5 (6.4–18.3)
1-year PFS: 39%
NR
Cabozantinib + nivolumab
(2022)(30)
II 40 32 (80) papillary
2 (5) translocation unspecified
6 (15) unclassified
ORR 47.5 (31.5–63.9) 12.5 (6.3–16.4) 28 (16.3–NE)
Nivolumab + ipilimumab (Checkmate 920, 2022)(31) IIIb/IV 52 18 (35) papillary
7 (13) chromophobe
1 (2) medullary
2 (4) collecting duct
2 (4) translocation, unspecified
22 (42) unclassified
Grade ≥3 immune-mediated adverse events 19.6 (9.4–33.9) 3.7 (2.7–4.6) 21.2 (16.6–NE)
Pembrolizumab + lenvatinib (KEYNOTE-B61, 2023)(33) II 158 93 (59) papillary
29 (18) chromophobe
6 (4) translocation
9 (6) other
21 (13) unclassified
ORR 49 (41–57) 18 (14–NR)
1-year PFS = 63%
NR
1-year OS = 82%

ORR: overall response rate, mPFS: median progression-free survival, OS: overall survival, NA: not assessed, NR: not reached, NE: not evaluated.