Table 4. In Vitro Mouse Metabolism of 1i, 2c, and 2ea.
| compound | liver microsomes CLint (mL/min/kg) | S9 fraction CLint (mL/min/kg) | hepatocytes CLint (mL/min/kg) |
|---|---|---|---|
| 1i | <24 | 0 | 143 |
| 2c | <24 | 1 | 132 |
| 2e | 27 | 4 | 69 |
Compounds quantified by LC-MS at five time points over 5 h, n = 1.