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. 2023 Oct 3;13(10):1480. doi: 10.3390/biom13101480

Table 1.

A summary of the main current PARPi combination clinical trials.

Trial Name Combination Therapy Phase Cohort Start
Completion Date
Ref
PARPi + Chemotherapy (STUDY41)
NCT01081951
Olaparib + Paclitaxel + Carbopatin II Platinum sensitive advanced ovarian cancer 4 Feb 2010–
29 Dec 2023
[59]
PARPi + Immunotherapy (TOPACIO)
NCT02657889
Niraparib + Pembrolizumab II Platinum-resistance ovarian cancer (regardless BRCA or HRD status) or BRCA mutated metastatic TNBC 15 Apr 2016–
17 Sep 2021
[66,67]
(ENGOT-OV44) NCT03602859 Niraparib + Dostarlimab III Stage III or IV nonmucinous Epithelial ovarin cancer 11 Oct 2018–
22 Jun 2026
[71]
(MEDIOLA)
NCT02734004
Olaparib + Durvalumab II gBRCAm platinum-sensitive ovarian cancer 28 Oct 2018–
2026
[68]
(OPEB-1)
NCT04361370
Olaparib + Durvalumab + Bevacizumab II Platinum-sensitive recurrent BRCA wt ovarian cancer 28 Oct 2020–
Aug 2026
[70]
(ATHENA) NCT03522246 Rucaparib + Nivolumab III Newly diagonsed advanced (FIGO stage III-IV) epithelial ovarin cancer. Fallopian Tube diseases. 14 May 2018–
30 Dec2030
[72]
(DUO-O) NCT03737643 Olaparib + Durvalumab III Newly diagonsed advanced ovarain cancer (Regardless BRCA status) 4 Jan 2019–
25 May 2028
[73]
NCT02849496 Olaparib + Atezolizumb (Anti-PD-L1) II Locally advanced unresectable or metastatic non-HER2 positive breast cancer 30 Mar 2017–
31 Aug 2023
[74]
PARPi +
Anti-angiogenic agents
NCT01116648 Olaparib + Cediranib I/II Relapsed Platinum sensitive high-grade or endometrioid ovarian cancer 25 Mar 2010–
31 Oct 2018
[75]
(NRG-GY005)
NCT02502266
Olaparib + Cediranib II/III Recurrent Platinum-resistant ovarian cancer, Fallopian Tube diseases. 3 May 2016–
30 Jun 2024
[76]
(PAOLA-1)
NCT02477644
Olaparib + Bevacizumab III HRD positive high-grade ovarian cancer 6 May 2015–
22 Mar 2022
[77,78,79]
NCT02354131 Niraparib + Bevacizumab I/II platinum-sensitive ovarian cancer 15 Feb 2015–
15 Dec 2021
[80]
PARPi + PI3K/AKT pathway inhibitors NCT01623349 Olaparib + Alpelisib I Platinum-resistant ovarian cancer or recurrent triple negative breast cancer (regardless BRCA or HRD status) Sep 2012–
Dec 2020
[81,82]
(EPIK-O)
NCT04729387
Olaparib + Alpelisib III Platinum-resistant or refractory high-grade serious epithelial ovarian cancer (HGSOC) with BRCA wt. 2 Jul 2021–
29 Jul 2025
[83]
NCT02208375 Olaparib + Vistusertib or Olaparib + Capivasertib I/II Recurrent endometrial, triple negative breast cancer or ovarian cancer 11 Nov 2014–
20 Jun 2024
[84]
NCT02338622 Olaparib + Capivasertib I Platinum-resistant HGSOC (regardless BRCA or HRD status) 31 Mar 2014–
21 Mar 2017
[85]
NCT03586661 Niraparib + Copanlisib I Recurrent high-grade serous or BRCA mutant ovarian cancer 29 Apr 2019–
31 Dec 23
[86]
PARPi + MAPK pathway inhibitors NCT03162627 Olaprib + Selumetinib I/II PARPi resistant ovarian cancer or Solid tumor with RAS pathway alteration 4 Aug 2017–
30 Aug 2026
[87]
PARPi + Epigenetic drugs NCT02878785 Talazoparib + Decitabine I/II Acute Myeloid Leukemia Aug 2016–
19 Nov 2020
[88]
NCT03742245 Olaprib + Vorinostat I Relapsed metastatic breast cancer 11 Jun 2019–
1 Sep 2024
[89]
PARPi + DDR inhibitors (CAPRI) NCT03462342 Olaparib + Ceralasertib II Platinum-resistant HGSOC 9 Mar 2018–
31 Dec 2023
[90]
NCT04267939 Niraparib + Elimsertib I Recurrent advanced solid tumors and ovarian cancer. 26 Feb 2020–
3 Mar 2025
[91]
NCT03057145 Olaparib + Prexasertib I BRCA mutant PARPi resistant HGSOC 10 Mar 2017–
9 Jun 2021
[92]
(EFFORT)
NCT03579316
Olaparib + Adavosertib II PARPis resistant ovarian cancer 7 Dec 2018–
30 Dec 2023
[93]
NCT04991480 Talozoparib + ART4215 I/II BRCA deficient breast cancer 13 Sep 2021–
Aug 2025
[94]