Table 3. PDE Selectivitya.
cpd | PDE3A | PDE4D3 | PDE5A | PDE6C | PDE10A |
---|---|---|---|---|---|
14b | 0 | 1.1 | 9.7 | 13.5 | 13.8 |
14c | 0.8 | 6 | 36 | 20 | 18 |
18a | 3 | 8 | 61 | 30 | 2 |
18d | 0 | 0 | 48 | 12 | 5 |
23b | 2 | 8 | 20 | 7 | 8 |
% inhibition at 500 nM, average of three independent determinations.