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. 2023 Oct 13;9(11):2141–2159. doi: 10.1021/acsinfecdis.3c00250

Table 1. Compounds 11 and 13 Display Enhanced Antibacterial Activity against S. aureus and S. epidermidis.

    minimum inhibitory concentration (μg/mL)
strain 1771 9 10 11 12 13 14
S. aureus
LAC 8 32–64 64 4 8 0.5 >64
MW2 8 64 64 2 8 0.5 >64
Newman 4–8 32 64 2 8 0.5 >64
SH1000 4–8 32 64 2 8 0.5 >64
MRSA252 8 64 64 4 16 1 >64
TW20 8 32 64 2 8 0.5 >64
Mu50 4–8 64 64 2 4–8 0.5 >64
Mu3 8–16 64 64 2 8 0.5 >64
EMRSA-15 8–16 64 32–64 2 8 0.5 >64
S. epidermidis
RP62A 8–16 32 64 2–4 4–8 0.5 >64
311 8–16 64 32–64 2 4–8 0.5 >64
771 8–16 64 32–64 2 4–8 0.5 >64
780 8–16 32 32–64 4 4–8 0.5–1 >64
319 8–16 64 64 2 4–8 1 >64
322 16 64 64 4 8 0.5 >64
305 8–16 64 32–64 2–4 8 0.5–1 >64