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. 2023 Oct 13;9(11):2141–2159. doi: 10.1021/acsinfecdis.3c00250

Table 2. Compound 13 Displays Enhanced Activity against Other Gram-Positive Species.

  MIC (μg/mL)
bacterial species (strain) 1771 13
B. subtilis (W168) 4–8 0.5–1
E. faecalis (JH2-2) 16 2
E. faecium (C68) >128 >128
S. pyogenes (NCTC 8198) 32–64 16–32
S. pyogenes (NCTC 12048) 128 64
S. agalactiae (18R521) 128 64
S. agalactiae (COH1) >128 128
S. dysgalactiae (NCTC 13762) 128 64
S. dysgalactiae (NCTC 10238) >128 64