Table 1. Pharmacokinetic Parameters of Intravenously and Orally Administered Enoxaparin with and without Cellulose–Mercaptosuccinate.
| dose (mg/kg) | AUC0–8 (μg/mL h) | Cmax (IU/mL) | Tmax (h) | bioavailability (%) | |
|---|---|---|---|---|---|
| enoxaparin i.v. | 0.2 | 15.22 | 0.62936 | 0 | |
| enoxaparin oral | 10 | 5.45 | 0.04576 | 2 | 0.72 |
| enoxaparin + cellulose–mercaptosuccinate oral | 10 | 68.36 | 0.24058 | 1 | 8.98 |