Skip to main content
. 2023 Nov 23;13(49):34348–34357. doi: 10.1039/d3ra05942a

Prediction of binding free energy (kcal mol−1 ± average standard error) using MM-PBSA and MM-GBSA.

Component of energy COX-2:LUR COX-2:RDUE2 COX-2:SDT29
ΔEvdW −36.542 ± 0.185 −44.053 ± 0.200 −44.092 ± 0.217
ΔEele −42.044 ± 0.488 −30.286 ± 0.710 −48.408 ± 0.535
ΔGeleGB 50.039 ± 0.432 49.963 ± 0.588 64.917 ± 0.480
ΔGsolvGB 44.701 ± 0.431 43.840 ± 0.586 58.964 ± 0.478
ΔGbindGB −33.888 ± 0.160 −30.498 ± 0.243 −33.536 ± 0.242
ΔGelePB 47.850 ± 0.495 54.224 ± 0.653 66.261 ± 0.477
ΔGsolvPB 42.879 ± 0.497 48.318 ± 0.654 60.171 ± 0.477
ΔGbindPB −35.710 ± 0.277 −26.021 ± 0.323 −32.329 ± 0.317