Table 5.
Cells | Incubation Time (h) | Molar Activity (MBq/nmol) | |||||||
---|---|---|---|---|---|---|---|---|---|
1.1 | 1.3 | 2.3 | 5.4 | 7.9 | 13.7 | 15.3 | 38.3 | ||
AR42J uptake (%) | 1 | 0.4 ± 0.1 | 4.1 ± 0.2 | 4.2 ± 0.0 | 2.6 ± 0.2 | 7.5 ± 0.4 | |||
24 | 0.6 ± 0.0 | 8.6 ± 0.5 | 9.1 ± 0.4 | 4.9 ± 0.6 | 13.6 ± 0.2 | ||||
48 | 17.9 ± 0.7 | ||||||||
72 | 16.5 ± 1.3 | ||||||||
HEK293 sst2 uptake (%) | 1 | 1.2 ± 0.3 | 1.3 ± 0.1 | 3.9 ± 0.2 | 1.6 ± 0.3 | 2.1 ± 0.1 | 2.8 ± 0.1 | 1.2 ± 0.3 | |
24 | 2.6 ± 0.6 | 1.0 ± 0.0 | 2.8 ± 0.2 | 4.0 ± 0.3 | 4.3 ± 0.2 | 4.3 ± 0.9 | 2.6 ± 0.6 |