Table 6.
Cells | Incubation Time (h) | Molar Activity (MBq/nmol) | |||||||
---|---|---|---|---|---|---|---|---|---|
0.2 | 0.8 | 1.0 | 3.3 | 3.8 | 5.2 | 13.9 | 15.5 | ||
AR42J uptake (%) | 1 | 0.8 ± 0.1 | 1.4 ± 0.1 | 1.5 ± 0.1 | n.d. | 3.8 ± 0.2 | 5.3 ± 0.3 | 4.6 ± 0.3 | |
24 | 2.6 ± 0.2 | 4.4 ± 0.4 | 4.5 ± 0.0 | 8.0 ± 1.0 | 1.5 ± 0.1 | 8.7 ± 0.7 | 17.0 ± 0.7 | ||
48 | 3.2 ± 0.4 | 3.1 ± 0.1 | 9.6 ± 0.7 | ||||||
72 | 5.2 ± 0.4 | 25.0 ± 0.5 | |||||||
HEK293 sst2 uptake (%) | 1 | 5.1 ± 0.5 | |||||||
24 | 4.0 ± 0.5 | ||||||||
48 | 9.1 ± 0.5 | ||||||||
72 | 7.8 ± 0.0 |