BBB assay of key benzyloxy chalcone compounds using the PAMPA methoda.
| Compound | Experimental Pe (×10−6 cm s−1) | Prediction |
|---|---|---|
| ISB1 | 4.93 ± 0.13 | CNS+ |
| ISFB1 | 4.09 ± 0.24 | CNS+ |
| Selegiline | 5.69 ± 0.04 | CNS+ |
Pe (10−6 cm s−1) > 4.00: CNS+ (high permeation).
| Compound | Experimental Pe (×10−6 cm s−1) | Prediction |
|---|---|---|
| ISB1 | 4.93 ± 0.13 | CNS+ |
| ISFB1 | 4.09 ± 0.24 | CNS+ |
| Selegiline | 5.69 ± 0.04 | CNS+ |
Pe (10−6 cm s−1) > 4.00: CNS+ (high permeation).