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. Author manuscript; available in PMC: 2023 Dec 8.
Published in final edited form as: J Med Chem. 2021 Oct 14;64(20):15334–15348. doi: 10.1021/acs.jmedchem.1c01370

Table 3.

The IC50 Values of the Advanced Compounds

inhibitors molecular weight IC50 (μM)a
CC10501 204 181 ± 40
RU-NT-70 281 19 ± 5
RU-NT-75 246 48 ± 11
RU-NT-93 232 14 ± 3
RU-NT-102 232 15 ± 3
a

The IC50 values were determined in vitro by qRT-PCR using yeast ribosomes as described in Figure 8.