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. 2023 Nov 20;71(48):18674–18684. doi: 10.1021/acs.jafc.3c06300

Table 2. BLCFA Exert Cytotoxicity to Cancer Cells in Vitro and in Vivo.

BLCFA cancer types in vitro or in vivo animal model cell lines dosage treatment period ref
iso-15:0 prostate cancer in vivo MetaMouse orthotopic model   35, 70, and 105 mg/kg/day 43 days (61)
iso-15:0 prostate cancer in vitro   DU 145 0–60 μg/mL 48 h (61)
anteiso-15:0 prostate cancer in vitro   DU 145, PC3 0–120 μg/mL 72 h (65)
iso-15:0 liver cancer in vivo MetaMouse orthotopic model   70 mg/kg/day 40 days (61)
iso-15:0 Liver cancer in vitro   SNU-423 0–60 μg/mL 48 h (61)
iso-15:0 T-cell non-Hodgkin lymphomas in vivo BALB/c nude mice   70 mg/kg/day 15 days in EL4 cell xenografts; 30 days in Jurkat cell xenografts (60)
iso-15:0 T-cell non-Hodgkin lymphomas in vitro   Jurkat, Hut78, and EL4 0–80 μg/mL 24, 48, and 72 h (60)
iso-15:0 bladder cancer in vitro   T24, 5637, and UM-UC-3 0–140 μg/mL 12 and 24 h (62)
iso-15:0 leukemia in vitro   K-562 0–60 μg/mL 48 h (61)
iso-15:0 colon cancer in vitro   HCT 116 0–60 μg/mL 48 h (61)
iso-15:0 small cell lung cancer in vitro   NCI-H1688 0–60 μg/mL 48 h (61)
anteiso-15:0 nonsmall cell lung cancer in vitro   A549 0–120 μg/mL 72 h (65)
anteiso-15:0 nonsmall cell lung cancer in vitro   H1299 0–120 μg/mL 72 h (65)
iso-15:0 pancreatic cancer in vitro   BxPC-3 0–60 μg/mL 48 h (61)
iso-15:0 gastric cancer in vitro   NCI-SNU-1 0–60 μg/mL 48 h (61)
iso-15:0 breast cancer in vitro   MCF7 0–60 μg/mL 48 h (61)
iso-15:0 breast cancer in vitro   MCF7 50–400 μM 24, 48, and 72 h (52)
anteiso-15:0 breast cancer in vitro   MCF-7 0–120 μg/mL 72 h (65)
iso-15:0 breast cancer in vitro   SKBR-3 0.05–0.2 mM 24 h (63)
iso-15:0 breast cancer in vitro   SKBR-3 0–1 mM 72 h (64)
iso-17:0 breast cancer in vitro   MCF7 50–400 μM 24, 48, and 72 h (52)