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. 2023 Nov 15;66(23):15629–15647. doi: 10.1021/acs.jmedchem.3c01233

Table 3. Diamino-cyclopentane Stereochemical Comparison against CDK9/Cyclin T1.

graphic file with name jm3c01233_0016.jpg

a

Enzymatic assay conducted at 10 μM ATP concentration (CDK9/cyclin T1 at Km).