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. 2023 Dec 14;66(24):16704–16727. doi: 10.1021/acs.jmedchem.3c01406

Table 1. Biochemical Efficacy, Potency, and Affinity of Compounds 1–9.

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a

Means derived from fitting concentration-response data from the coupled enzyme assay performed in triplicate.

b

Means derived from fitting concentration-response data from the coupled enzyme assay performed in triplicate.

c

Means derived from the FP displacement assay performed in triplicate.